Abstract

Saponins are glycosides with triterpenoid or spirostane aglycones that demonstrate various pharmacological effects against mammalian diseases. To promote the research and development of anticancer agents from saponins, this review focuses on the anticancer properties of several typical naturally derived triterpenoid saponins (ginsenosides and saikosaponins) and steroid saponins (dioscin, polyphyllin, and timosaponin) isolated from Chinese medicines. These saponins exhibit in vitro and in vivo anticancer effects, such as anti-proliferation, anti-metastasis, anti-angiogenesis, anti-multidrug resistance, and autophagy regulation actions. In addition, related signaling pathways and target proteins involved in the anticancer effects of saponins are also summarized in this work.

Details

Title
Saponins from Chinese Medicines as Anticancer Agents
Author
Xu, Xiao-Huang; Li, Ting; Fong, Chi Man Vivienne; Chen, Xiuping; Chen, Xiao-Jia; Wang, Yi-Tao; Huang, Ming-Qing; Lu, Jin-Jian
First page
1326
Publication year
2016
Publication date
2016
Publisher
MDPI AG
e-ISSN
14203049
Source type
Scholarly Journal
Language of publication
English
ProQuest document ID
1831823844
Copyright
Copyright MDPI AG 2016